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TM-score TM-align US-align MM-align RNA-align NW-align LS-align EDTSurf MVP MVP-Fit SPICKER HAAD PSSpred 3DRobot MR-REX I-TASSER-MR SVMSEQ NeBcon ResPRE TripletRes DeepPotential WDL-RF ATPbind DockRMSD DeepMSA FASPR EM-Refiner GPU-I-TASSER

BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameAlpha-2C adrenergic receptor
SpeciesDidelphis virginiana (North American opossum)
GeneADRA2C
SynonymAlpha-2C adrenoceptor
Alpha-2C adrenoreceptor
Alpha-2CAR
DiseaseN/A for non-human GPCRs
Length469
Amino acid sequenceMDLQLTTNSTDSGDRGGSSNESLQRQPPSQYSPAEVAGLAAVVSFLIVFTIVGNVLVVIAVLTSRALKAPQNLFQVSLASADILVATLVMPFSLANELMNYWYFGKVWCVIYLALDVLFCTSSIVHLCAISLDRYWSVTQAVEYNLKRTPRRIKGIIVTVWLISAVISFPPLISLYRDPEDDLYPQCELNDETWYILSSCIGSFFAPCIIMVLVYVRIYRVAKLRTRTLSEKRTVPEGSSQTENGLSRPPVGAGPSTAAAAAASLRLQAGENGHYHLHHHHHHLHHHHHHHHHQLRKSAELEDIELEESSTSENRRRRRSREEAAARKGSRGFSFSFSSTKGGQSAGAGSRLSRASNRSLEFFSTHRRRKRSSLCRRKVTQAREKRFTFVLAVVMGVFVVCWFPFFFTYSLYGICREACQVPETLFKFFFWIGYCNSSLNPVIYTIFNQDFRRSFKHILFKKKKKTSLQ
UniProtP35405
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLN/A
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 11
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
266172D structureYohimbineC21H26N2O3354.454 / 22.9Yes
1208162D structureIDAZOXANC11H12N2O2204.2293 / 10.7Yes
1231792D structureAtipamezoleC14H16N2212.2961 / 13.0Yes
1313742D structureprazosinC19H21N5O4383.4088 / 12.0Yes
1608522D structureSpiroxatrineC22H25N3O3379.465 / 13.1Yes
2122172D structureAC1NKXXYC17H19N3O281.3592 / 23.3Yes
2491022D structureD0V8NSC25H30N2O3406.5265 / 04.2Yes
3350032D structure(S)-mianserinC18H20N2264.3722 / 03.4Yes
3464702D structureSCHEMBL8097715C25H27NO5421.4936 / 14.4Yes
3857652D structureoxymetazolineC16H24N2O260.3812 / 22.9Yes
4340612D structurechlorpromazineC17H19ClN2S318.8633 / 05.2No

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