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GPCR

NameC-C chemokine receptor type 10
SpeciesHomo sapiens (Human)
GeneCCR10
SynonymCCR-10
CCR10
CC-CKR-10
G-protein coupled receptor 2
GPR-2
[ Show all ]
DiseaseInflammatory disease
Length362
Amino acid sequenceMGTEATEQVSWGHYSGDEEDAYSAEPLPELCYKADVQAFSRAFQPSVSLTVAALGLAGNGLVLATHLAARRAARSPTSAHLLQLALADLLLALTLPFAAAGALQGWSLGSATCRTISGLYSASFHAGFLFLACISADRYVAIARALPAGPRPSTPGRAHLVSVIVWLLSLLLALPALLFSQDGQREGQRRCRLIFPEGLTQTVKGASAVAQVALGFALPLGVMVACYALLGRTLLAARGPERRRALRVVVALVAAFVVLQLPYSLALLLDTADLLAARERSCPASKRKDVALLVTSGLALARCGLNPVLYAFLGLRFRQDLRRLLRGGSCPSGPQPRRGCPRRPRLSSCSAPTETHSLSWDN
UniProtP46092
Protein Data BankN/A
GPCR-HGmod modelP46092
3D structure modelThis predicted structure model is from GPCR-EXP P46092.
BioLiPN/A
Therapeutic Target DatabaseT71054
ChEMBLCHEMBL2321628
IUPHAR67
DrugBankN/A

Known ligands

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Total entries: 127
Page:  / 2 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
5214472D structureCHEMBL3731686C27H26Cl2FN7O4S634.5088 / 34.7No
5359542D structureCHEMBL3959737C21H25Cl2N5O3S498.4236 / 23.6Yes
5215182D structureCHEMBL3727384C27H26Cl2FN7O4S634.5088 / 34.7No
5360422D structureCHEMBL3923733C23H27N5O3S453.5615 / 22.6Yes
5216032D structureCHEMBL3733065C29H30FN7O5S607.6619 / 32.9No
5361512D structureCHEMBL3919363C20H24Cl2N6O3S499.4117 / 22.7Yes
5217422D structureCHEMBL3729731C29H30FN7O5S607.6619 / 32.9No
5219242D structureCHEMBL3732878C28H28ClFN6O3S583.0798 / 25.1No
5220142D structureCHEMBL3730003C28H26ClFN6O4S597.0628 / 24.4No
5364912D structureCHEMBL3960700C22H25N5O4S455.5336 / 31.2Yes
5223142D structureCHEMBL3731390C30H29ClN6O5S621.1098 / 23.7No
5224032D structureCHEMBL3731840C25H23Cl2FN6O4S593.4559 / 24.8No
5534152D structureeut-22C23H27N5O3S453.5615 / 22.6Yes
5367812D structureCHEMBL3889627C23H27N5O3S453.5615 / 22.6Yes
5225942D structureCHEMBL3728353C29H29FN6O5S592.6469 / 23.2No
5369852D structureCHEMBL3943972C18H24Cl2N6O3S475.3897 / 22.6Yes
5227262D structureCHEMBL3728979C27H24F4N6O4S604.58111 / 24.8No
5370392D structureCHEMBL3948828C19H25Cl2N5O3S474.4016 / 22.6Yes
5370452D structureCHEMBL3971886C23H27N5O3S453.5615 / 22.6Yes
5229392D structureCHEMBL3728246C25H21Cl2FN6O4S591.4398 / 24.6No
5229622D structureCHEMBL3729606C28H28ClF2N7O4S632.0849 / 34.6No
5229782D structureCHEMBL3728616C27H28ClFN6O4S587.0679 / 24.0No
5232362D structureCHEMBL3731147C30H32FN7O5S621.6889 / 23.3No
5232682D structureCHEMBL3728071C28H23Cl2FN8O3S641.50310 / 24.6No
5235072D structureCHEMBL3731775C30H29ClN6O5S621.1098 / 23.7No
5237002D structureCHEMBL3731933C29H29FN6O5S592.6469 / 23.2No
5238402D structureCHEMBL3732508C30H29FN6O5S604.6579 / 23.1No
5238682D structureCHEMBL3728121C29H29ClN6O5S609.0988 / 23.7No
5240142D structureCHEMBL3731832C32H34ClN7O6S680.1779 / 34.0No
5381372D structureCHEMBL3909737C23H27N5O3S453.5615 / 22.6Yes
5489322D structureCHEMBL3932155C19H24Cl2N6O5S519.3988 / 22.5No
5489332D structureCHEMBL3908983C19H24Cl2N6O5S519.3988 / 22.5No
5381932D structureCHEMBL3908230C19H24Cl2N6O5S519.3988 / 22.5No
5241272D structureCHEMBL3731438C28H30FN7O4S579.6518 / 33.9No
5241672D structureCHEMBL3733165C28H23Cl2FN8O3S641.50310 / 24.9No
5382962D structureCHEMBL3942284C23H27N5O3S453.5615 / 22.6Yes
5242542D structureCHEMBL3728606C28H28ClFN6O4S599.0788 / 24.8No
5384002D structureCHEMBL3945769C24H29N5O3S467.5885 / 12.6Yes
5249872D structureCHEMBL3730752C26H23F3N6O4S572.56310 / 23.5No
5391492D structureCHEMBL3979967C19H24Cl3N5O3S508.8436 / 23.6No
5391912D structureCHEMBL3933303C23H31N5O3S457.5936 / 22.6Yes
5252112D structureCHEMBL3732652C28H30FN7O3S2595.7128 / 34.5No
5253042D structureCHEMBL3732876C29H30ClN7O5S624.1138 / 33.4No
5253272D structureCHEMBL3732868C26H23Cl2FN6O4S605.4668 / 24.6No
5253942D structureCHEMBL3729178C28H28ClFN8O4S627.0929 / 33.7No
5255002D structureCHEMBL3729146C27H27FN6O4S550.6098 / 23.7No
5255782D structureCHEMBL3731219C27H25Cl2FN6O4S619.4938 / 25.0No
5256052D structureCHEMBL3727497C28H27ClFN7O4S612.0779 / 24.0No
5257092D structureCHEMBL3732344C28H25ClF4N6O4S653.0511 / 25.3No
5497972D structureCHEMBL3928968C19H21Cl2N5O3S470.3696 / 22.3Yes
5498122D structureCHEMBL3950532C18H24Cl2N6O3S475.3897 / 22.1Yes
5398792D structureCHEMBL3969321C20H23Cl2N5O3S484.3966 / 22.6Yes
5259402D structureCHEMBL3728332C28H30FN7O4S579.6519 / 33.3No
5261772D structureCHEMBL3731138C29H30N6O4S558.6577 / 23.6No
5262982D structureCHEMBL3730468C28H29FN6O5S580.6359 / 23.5No
5264352D structureCHEMBL3729372C27H28F2N6O3S554.6179 / 24.3No
5265232D structureCHEMBL3727981C26H27FN6O5S2586.65710 / 23.4No
5268042D structureCHEMBL3732672C27H26ClF2N7O4S618.0579 / 34.2No
5268232D structureCHEMBL3732501C27H28ClFN6O3S571.0688 / 24.9No
5268632D structureCHEMBL3730497C28H31N7O4S561.6617 / 33.3No
5502452D structureCHEMBL3973467C18H24Cl2N6O3S475.3897 / 22.4Yes
5271552D structureCHEMBL3731456C28H26ClF2N7O4S630.0689 / 35.0No
5503112D structureCHEMBL3964878C22H27Cl2N3O3S484.4365 / 24.6Yes
5410682D structureCHEMBL3926111C22H27Cl2N3O3S484.4365 / 24.6Yes
5503292D structureCHEMBL3979899C19H21N5O3S399.4695 / 21.4Yes
5272882D structureCHEMBL3728893C29H29F2N7O4S609.6539 / 34.7No
5504192D structureCHEMBL3900672C17H19Cl2N5O3S444.3316 / 21.8Yes
5274632D structureCHEMBL3728376C27H27ClFN7O4S600.0668 / 34.1No
5415242D structureCHEMBL3975141C25H28N4O3S464.5845 / 13.8Yes
5277622D structureN-[7-(4-fluoro-2-methylphenylamino)-6-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-3-ylsulfonyl]cyclopropanecarboxamideC29H29FN6O4S576.6478 / 24.1No
5282222D structureCHEMBL3728115C27H28ClN7O4S582.0767 / 34.0No
5423372D structureCHEMBL3951650C20H24Cl2N6O3S499.4117 / 22.4Yes
5286702D structureCHEMBL3733183C26H21Cl2FN8O3S2647.52511 / 25.1No
5287302D structureCHEMBL3732275C29H27Cl2FN6O5S661.539 / 24.5No
5426842D structureCHEMBL3890608C23H27N5O3S453.5615 / 22.6Yes
5289712D structureCHEMBL3733316C26H25ClN6O5S569.0338 / 24.2No
5290492D structureCHEMBL3731999C32H30FN7O4S627.6958 / 35.6No
5429892D structureCHEMBL3971826C22H25N5O3S439.5345 / 22.2Yes
5290962D structureCHEMBL3729920C26H23Cl2FN6O4S605.4668 / 24.6No
5290972D structureCHEMBL3728619C27H26ClF2N7O4S618.0579 / 34.2No
5292722D structureCHEMBL3728998C26H25ClFN7O4S586.0398 / 33.7No
5296192D structureCHEMBL3731666C28H30FN7O3S563.6528 / 14.1No
5296932D structureCHEMBL3727493C27H25F5N6O3S608.58812 / 25.1No
5298382D structureCHEMBL3728415C28H30N6O5S562.6458 / 24.3No
5300212D structureCHEMBL3730157C28H28ClFN6O4S599.0788 / 24.8No
5442632D structureCHEMBL3940706C20H26Cl2N4O3S473.4135 / 23.0Yes
5443272D structureCHEMBL3964547C19H24Cl3N5O3S508.8436 / 23.3No
5304072D structureCHEMBL3733128C27H27FN6O5S566.6089 / 33.0No
5304452D structureCHEMBL3732824C29H26Cl2N6O5S641.5248 / 23.9No
5304562D structureCHEMBL3729504C27H25F3N6O4S586.5910 / 24.0No
5304572D structureCHEMBL3727436C28H29ClFN7O4S614.0938 / 34.5No
5446812D structureCHEMBL3955499C21H25Cl2N5O3S498.4236 / 23.1Yes
5307032D structureCHEMBL3731872C29H27ClF2N6O4S629.089 / 24.8No
5448392D structureCHEMBL3946799C21H22Cl2F3N5O3S552.3949 / 23.7No
5520252D structureCHEMBL3944089C19H25Cl2N5O3S474.4016 / 22.4Yes
5308612D structureCHEMBL3732278C28H27ClN6O5S595.0718 / 23.2No
5309432D structureCHEMBL3731105C28H28F2N6O4S582.6279 / 24.2No
5310092D structureCHEMBL3732825C28H26ClFN6O5S613.0619 / 23.4No
5451632D structureCHEMBL3891692C23H24F3N5O3S507.5328 / 23.2No
5452622D structureCHEMBL3891289C22H26Cl3N3O3S518.8785 / 25.2No

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