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GPCR

NameGrowth hormone-releasing hormone receptor
SpeciesHomo sapiens (Human)
GeneGHRHR
Synonymgrowth hormone-releasing factor receptor
GRFR
GRF receptor
GHRH receptor
Ghrfr
DiseaseN/A
Length423
Amino acid sequenceMDRRMWGAHVFCVLSPLPTVLGHMHPECDFITQLREDESACLQAAEEMPNTTLGCPATWDGLLCWPTAGSGEWVTLPCPDFFSHFSSESGAVKRDCTITGWSEPFPPYPVACPVPLELLAEEESYFSTVKIIYTVGHSISIVALFVAITILVALRRLHCPRNYVHTQLFTTFILKAGAVFLKDAALFHSDDTDHCSFSTVLCKVSVAASHFATMTNFSWLLAEAVYLNCLLASTSPSSRRAFWWLVLAGWGLPVLFTGTWVSCKLAFEDIACWDLDDTSPYWWIIKGPIVLSVGVNFGLFLNIIRILVRKLEPAQGSLHTQSQYWRLSKSTLFLIPLFGIHYIIFNFLPDNAGLGIRLPLELGLGSFQGFIVAILYCFLNQEVRTEISRKWHGHDPELLPAWRTRAKWTTPSRSAAKVLTSMC
UniProtQ02643
Protein Data Bank2xdg
GPCR-HGmod modelQ02643
3D structure modelThis structure is from PDB ID 2xdg.
BioLiPBL0126345,BL0126346
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL2032
IUPHARN/A
DrugBankBE0000625

Known ligands

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Total entries: 3
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
5501772D structureGHRH(1-44)C216H360N72O63S5005.7672 / 81-23.2No
4571042D structureDocetaxel trihydrateC43H59NO17861.93517 / 8N/ANo
4260712D structuredocetaxelC43H53NO14807.8914 / 51.6No

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