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TM-score TM-align US-align MM-align RNA-align NW-align LS-align EDTSurf MVP MVP-Fit SPICKER HAAD PSSpred 3DRobot MR-REX I-TASSER-MR SVMSEQ NeBcon ResPRE TripletRes DeepPotential WDL-RF ATPbind DockRMSD DeepMSA FASPR EM-Refiner GPU-I-TASSER

BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameAdenosine receptor A3
SpeciesCanis lupus familiaris (Dog)
GeneADORA3
SynonymN/A
DiseaseN/A for non-human GPCRs
Length314
Amino acid sequenceMAVNGTALLLANVTYITVEILIGLCAIVGNVLVIWVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVISLGITIQFYNCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYRRVTTQRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEHQRNVTFLSCQFSSVMRMDYMVYFSFFTWILIPLVVMCAIYLDIFYVIRNKLNQNFSSSKETGAFYGREFKTAKSLFLVLFLFAFSWLPLSIINCITYFHGEVPQIILYLGILLSHANSMMNPIVYAYKIKKFKETYLLIFKTYMICQSSDSLDSSTE
UniProtQ28309
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL3611963
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 5
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GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
4687412D structureCHEMBL3612932C22H23ClN6O3S486.9758 / 42.5Yes
4714052D structureCHEMBL3612940C22H22ClN5O3S471.967 / 42.3Yes
4715302D structureCHEMBL3612939C21H20ClN5O3S457.9337 / 42.0Yes
4974462D structureCHEMBL3612931C21H21ClN6O3S472.9488 / 42.0Yes
5007522D structureCHEMBL3407784C20H19ClN6O3S458.9218 / 41.7Yes

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