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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameG-protein coupled bile acid receptor 1
SpeciesRattus norvegicus (Rat)
GeneGpbar1
SynonymBG37
Membrane-type receptor for bile acids
M-BAR
hGPCR19
GPR131
[ Show all ]
DiseaseN/A for non-human GPCRs
Length329
Amino acid sequenceMMSHNTTELSAIPRGVQELSLVLASLIVIANLLLALGIVLDRHLRSPPAGCFFLSLLLAGLLTGLALPTLPGLWNRSHQGYWSCLLLHLAPNFCFLSLLANLLLVHGERYMAVLQPLRPHGSVRLALFLTWISSLLFASLPALGWNHWSPGANCSSQAIFPAPYLYLEVYGLLLPAVGATALLSVRVLATAHHQLREIRRLERAVCRDAPSTLARALTWRQARAQAGATLLFLLCWGPYVATLLLSVLAYERRPPLGPVTLLSLISLGSASAAVVPVAMGLGDQRYTAPWRTAAQRWLQVLRGRPKRANPGPSTAYHSSSQCSTDLDLN
UniProtQ80T02
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL1075223
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 3
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
351382D structureCHEMBL2331646C22H29N5O2395.5075 / 22.5Yes
1327912D structureTGR5 Receptor AgonistC18H14Cl2N2O2361.2223 / 04.7Yes
3806712D structureCHEMBL576138C19H16Cl2N2O2375.2493 / 05.1No

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